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Study of G protein-coupled receptors dimerization: From bivalent ligands to drug-like small molecules

Mingcheng Qian, Zhengyang Sun, Xin Chen, Serge Van Calenbergh

2023Bioorganic Chemistry10 citationsDOIOpen Access PDF

Topics & Concepts

Bivalent (engine)ChemistryG protein-coupled receptorReceptorMonomerSmall moleculeAffinitiesDrugBiophysicsStereochemistryMoleculeCombinatorial chemistryBiochemistryPharmacologyMetalBiologyPolymerOrganic chemistryReceptor Mechanisms and SignalingNeuropeptides and Animal PhysiologyChemical Synthesis and Analysis
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