Advancing targeted protein degrader discovery by measuring cereblon engagement in cells
Breanna L. Zerfas, Fidel Huerta, Hu Liu, Guangyan Du, Nathanael S. Gray, Lyn H. Jones, Radosław P. Nowak
Topics & Concepts
CereblonLuciferaseChemistryUbiquitin ligaseUbiquitinFusion proteinCell biologyBioluminescenceComputational biologyBiochemistryBiologyGeneRecombinant DNATransfectionProtein Degradation and InhibitorsUbiquitin and proteasome pathwaysPeptidase Inhibition and Analysis