Litcius/Paper detail

Synthesis of dolutegravir derivatives modified by 1,2,3-triazole structure and their anti-inflammatory activity in LPS-induced BV2 cells

Xixi Hou, Longfei Mao, Xuanwei Zhang, Xi Wang, Lan Wang, Jianji Wang, Lan Wang, Jianji Wang

2024Bioorganic & Medicinal Chemistry Letters13 citationsDOI

Topics & Concepts

ChemistryDolutegravirTriazoleStructure–activity relationshipIn vitroCombinatorial chemistryStereochemistryPharmacologyBiochemistryOrganic chemistryVirusVirologyBiologyViral loadMedicineAntiretroviral therapyClick Chemistry and ApplicationsHIV/AIDS drug development and treatmentSynthesis and biological activity
Synthesis of dolutegravir derivatives modified by 1,2,3-triazole structure and their anti-inflammatory activity in LPS-induced BV2 cells | Litcius