Novel approach of multi-targeted thiazoles and thiazolidenes toward anti-inflammatory and anticancer therapy—dual inhibition of COX-2 and 5-LOX enzymes
Jaismy Jacob P, S. L. Manju
Topics & Concepts
ChemistryZileutonPharmacologyPharmacophoreArachidonate 5-lipoxygenaseCelecoxibEtoricoxibIn vivoCyclooxygenaseAnti-inflammatoryIC50ThiazolePotencyCarrageenanIn vitroEnzymeStereochemistryBiochemistryArachidonic acidMedicineOrganic chemistryBiotechnologyBiologyInflammatory mediators and NSAID effectsSynthesis and biological activitySynthesis and Reactions of Organic Compounds