Litcius/Paper detail

Design, synthesis, biological screening and molecular docking studies of novel multifunctional 1,4-di (aryl/heteroaryl) substituted piperazine derivatives as potential antitubercular and antimicrobial agents

Bruktawit Mekonnen Sanka, Dereje Mamo Tadesse, Endale Teju Bedada, Ephriem Mengesha, Neelaiah Babu G.

2021Bioorganic Chemistry16 citationsDOI

Topics & Concepts

ChemistryPiperazineDocking (animal)AntimicrobialArylStereochemistryCombinatorial chemistryLead compoundCytotoxicityProtein Data Bank (RCSB PDB)In vitroOrganic chemistryBiochemistryAlkylMedicineNursingSynthesis and biological activityCancer therapeutics and mechanismsQuinazolinone synthesis and applications