Litcius/Paper detail

Design, synthesis and molecular modeling of new quinazolin-4(3H)-one based VEGFR-2 kinase inhibitors for potential anticancer evaluation

Abdallah E. Abdallah, Sally I. Eissa, Maged Mohammed Saleh Al Ward, Reda R. Mabrouk, Ahmed B. M. Mehany, Mohamed Ayman El‐Zahabi

2021Bioorganic Chemistry69 citationsDOI

Topics & Concepts

ChemistryKinaseIC50Docking (animal)In vitroCell cultureThio-Tyrosine kinaseApoptosisCancer cellStereochemistryBiochemistryCombinatorial chemistryCancerSignal transductionBiologyNursingGeneticsMedicineQuinazolinone synthesis and applicationsHER2/EGFR in Cancer ResearchSynthesis and biological activity