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Recent advances in pyruvate dehydrogenase kinase inhibitors: Structures, inhibitory mechanisms and biological activities

Yiyang Li, Zhizhong Xie, Xiaoyong Lei, Xiaoyan Yang, Sheng Huang, Weixi Yuan, Xiangping Deng, Zhe Wang, Guotao Tang

2024Bioorganic Chemistry20 citationsDOI

Topics & Concepts

Cancer cellChemistryKinasePyruvate kinasePyruvate dehydrogenase complexGlycolysisBiochemistryPyruvate dehydrogenase kinaseEnzymeCancerOxidative phosphorylationCancer researchCell biologyBiologyGeneticsBiochemical Acid Research StudiesCancer, Hypoxia, and MetabolismATP Synthase and ATPases Research
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