Discovery of a series of 1H-pyrrolo[2,3-b]pyridine compounds as potent TNIK inhibitors
Bowen Yang, Qian Wu, Xia‐Juan Huan, Ying-Qing Wang, Yin Sun, Yueyue Yang, Tongchao Liu, Xin Wang, Lin Chen, Bing Xiong, Dongmei Zhao, Ze‐Hong Miao, Danqi Chen
Topics & Concepts
ChemistryPyridineDrug discoveryIC50Combinatorial chemistryPharmacologyStereochemistryBiochemistryIn vitroMedicinal chemistryBiologyMelanoma and MAPK PathwaysMechanisms of cancer metastasisCell death mechanisms and regulation