Synthesis, molecular docking and molecular dynamics studies of novel tacrine-carbamate derivatives as potent cholinesterase inhibitors
Özge Özten, Belma Zengin Kurt, Fatih Sönmez, Berna Doğan, Serdar Durdağı
Topics & Concepts
TacrineButyrylcholinesteraseChemistryAcetylcholinesteraseCarbamateCholinesteraseStereochemistryDocking (animal)AchéEnzymeSelectivityEnzyme inhibitorBiochemistryPharmacologyNursingMedicineCatalysisCholinesterase and Neurodegenerative DiseasesComputational Drug Discovery MethodsEnzyme function and inhibition