Novel sampangine derivatives as potent inhibitors of Cu2+-mediated amyloid-β protein aggregation, oxidative stress and inflammation
Xiaoyan Zou, Ren-ren Xie, Wěi Li, Chun-ling Su, Yu-si Chen, Huang Tang
Topics & Concepts
ChemistryIsothermal titration calorimetryProinflammatory cytokineOxidative stressChelationBlood–brain barrierCholinesteraseAcetylcholinesteraseMembrane permeabilityBiochemistryBiophysicsMembranePharmacologyInflammationEnzymeOrganic chemistryBiologyCentral nervous systemImmunologyNeuroscienceAlzheimer's disease research and treatmentsCholinesterase and Neurodegenerative DiseasesMedicinal Plants and Neuroprotection