The efflux pump ABCC1/MRP1 constitutively restricts PROTAC sensitivity in cancer cells
Gernot Wolf, Conner Craigon, Shao Thing Teoh, Patrick Essletzbichler, Svenja Onstein, Diane Cassidy, Esther C. H. Uijttewaal, Vojtech Dvorak, Yuting Cao, Ariel Bensimon, Ulrich Elling, Alessio Ciulli, Giulio Superti‐Furga
Topics & Concepts
EffluxABCC1Sensitivity (control systems)Cancer cellChemistryCell biologyCancerCancer researchBiologyMedicineBiochemistryInternal medicineGeneEngineeringTransporterATP-binding cassette transporterElectronic engineeringProtein Degradation and InhibitorsPeptidase Inhibition and AnalysisUbiquitin and proteasome pathways