Hydrazonoyl bromide precursors as DHFR inhibitors for the synthesis of bis-thiazolyl pyrazole derivatives; antimicrobial activities, antibiofilm, and drug combination studies against MRSA
Seham A. Ibrahim, Eman A. Fayed, Hala F. Rizk, Said E. Desouky, Ahmed Ragab
Topics & Concepts
AntimicrobialChemistryPyrazoleResazurinThiazoleBromideMinimum inhibitory concentrationMinimum bactericidal concentrationAntibioticsIC50Combinatorial chemistryStereochemistryIn vitroOrganic chemistryBiochemistrySynthesis and biological activityClick Chemistry and ApplicationsSynthesis and Biological Evaluation