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Exploration of the 2,3-dihydroisoindole pharmacophore for inhibition of the influenza virus PA endonuclease

Dominga Rogolino, Lieve Naesens, Jennifer Bartoli, Mauro Carcelli, Laura De Luca, Giorgio Pelosi, Ryjul W. Stokes, Ria Van Berwaer, Serena Vittorio, Annelies Stevaert, Seth M. Cohen

2021Bioorganic Chemistry13 citationsDOIOpen Access PDF

Topics & Concepts

PharmacophoreChemistryEndonucleasePolymeraseInfluenza A virusVirusDocking (animal)EnzymeRNA polymeraseBiochemistryVirologyRNABiologyGeneMedicineNursingInfluenza Virus Research StudiesRNA and protein synthesis mechanismsViral Infections and Immunology Research
Exploration of the 2,3-dihydroisoindole pharmacophore for inhibition of the influenza virus PA endonuclease | Litcius