Detection of Weak Organic Anion–Transporting Polypeptide 1B Inhibition by Probenecid with Plasma-Based Coproporphyrin in Humans
Yueping Zhang, Vinay K. Holenarsipur, Hamza Kandoussi, Jianing Zeng, T. Thanga Mariappan, Michael Sinz, Hong Shen
Topics & Concepts
ProbenecidOrganic anion transporter 1Organic anion-transporting polypeptideChemistryTransporterPharmacologyEndogenyKidneyPharmacokineticsIn vitroFurosemideEndocrinologyBiochemistryBiologyGeneOrganic chemistryDrug Transport and Resistance MechanismsPharmacological Effects and Toxicity StudiesHemoglobinopathies and Related Disorders