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Quantitative Investigation of Irinotecan Metabolism, Transport, and Gut Microbiome Activation

Md Masud Parvez, Abdul Basit, Parth B. Jariwala, Zsuzsanna Gáborik, Emese Kis, Scott Heyward, Matthew R. Redinbo, Bhagwat Prasad

2021Drug Metabolism and Disposition74 citationsDOIOpen Access PDF

Topics & Concepts

IrinotecanMetaboliteGlucuronidationPharmacologyMetabolismChemistryToxicityTransporterBiochemistryBiologyEnzymeMicrosomeCancerColorectal cancerOrganic chemistryGeneticsGeneCancer therapeutics and mechanismsDrug Transport and Resistance MechanismsAntibiotics Pharmacokinetics and Efficacy