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A Selective C–C Bond Cleavage Strategy Promoted by Visible Light

Rafael D. C. Gallo, M.T. Duarte, Amanda F. da Silva, Celso Y. Okada, Victor M. Deflon, Igor D. Jurberg

2021Organic Letters44 citationsDOIOpen Access PDF

Abstract

A new visible-light-promoted reaction between aryldiazoacetates and 1,3-diketones allows good yields and selectivities for C-C bond insertions, leading to the corresponding 1,4-dicarbonyl compounds. This transformation is straightforward and highly practical. It tolerates air and moisture and does not require the use of any metals. Mechanistic investigations support the involvement of a key cyclopropanol intermediate derived from an intramolecular rearrangement.

Topics & Concepts

ChemistryIntramolecular forceBond cleavagePhotochemistryCombinatorial chemistryCleavage (geology)Computational chemistryStereochemistryCatalysisOrganic chemistryGeotechnical engineeringFracture (geology)EngineeringCyclopropane Reaction MechanismsCatalytic C–H Functionalization MethodsRadical Photochemical Reactions
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