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Site-selective C–H alkylation of <i>myo</i>-inositol <i>via</i> organic photoredox catalysis

haonan cao, Tianyun Guo, Xuemei Deng, Xing Huo, Shouchu Tang, Jian Liu, Xiaolei Wang

2022Chemical Communications16 citationsDOI

Abstract

Site-selective photoredox reactions with aromatic olefins enable direct alkylation of unprotected myo -inositol at C4.

Topics & Concepts

AlkylationChemistryCatalysisInositolPhotoredox catalysisCombinatorial chemistryStereochemistryMedicinal chemistryOrganic chemistryBiochemistryPhotocatalysisReceptorSulfur-Based Synthesis TechniquesRadical Photochemical ReactionsCatalytic C–H Functionalization Methods
Site-selective C–H alkylation of <i>myo</i>-inositol <i>via</i> organic photoredox catalysis | Litcius