Discovery of dolutegravir-1,2,3-triazole derivatives against prostate cancer via inducing DNA damage
Shuyi Zhou, Xixi Hou, Ling Li, Lihao Guo, Huili Wang, Longfei Mao, Leilei Shi, Miaomiao Yuan
Topics & Concepts
DU145Prostate cancerDolutegravirCancer researchChemistryCancerPoly ADP ribose polymerasePharmacologyPolymeraseInternal medicineMedicineHuman immunodeficiency virus (HIV)VirologyDNABiochemistryLNCaPViral loadAntiretroviral therapyProstate Cancer Treatment and ResearchPARP inhibition in cancer therapyCancer Immunotherapy and Biomarkers