Medicinal chemistry perspective of JAK inhibitors: synthesis, biological profile, selectivity, and structure activity relationship
Lalmohan Maji, Sindhuja Sengupta, Gurubasavaraja Swamy Purawarga Matada, Ghanshyam Teli, G. Biswas, Pronoy Kanti Das, Manjunatha Panduranga Mudgal
Topics & Concepts
statJAK-STAT signaling pathwayRuxolitinibCancer researchJanus kinaseMedicineSignal transductionCytokineBiologyImmunologySTAT3Cell biologyTyrosine kinaseBone marrowMyelofibrosisCytokine Signaling Pathways and InteractionsChronic Lymphocytic Leukemia ResearchQuinazolinone synthesis and applications