Advances and perspectives of proteolysis targeting chimeras (PROTACs) in drug discovery
Jiayue Xi, Ruyue Zhang, Ke Chen, Lin Yao, Muqiong Li, Ru Jiang, Xiaoye Li, Li Fan
Topics & Concepts
Ubiquitin ligaseDrug discoveryChemistryProteasomeProteolysisLinkerComputational biologyUbiquitinBiologyBiochemistryComputer scienceEnzymeGeneOperating systemProtein Degradation and InhibitorsUbiquitin and proteasome pathwaysPeptidase Inhibition and Analysis