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Discovery of 7H-pyrrolo[2,3-d]pyridine derivatives as potent FAK inhibitors: Design, synthesis, biological evaluation and molecular docking study

Ruifeng Wang, Xiangxin Zhao, Sijia Yu, Yixuan Chen, Hengxian Cui, Tianxiao Wu, Chenzhou Hao, Dongmei Zhao, Maosheng Cheng

2020Bioorganic Chemistry28 citationsDOI

Topics & Concepts

ChemistryDocking (animal)IC50KinaseTyrosine kinaseCytotoxicityApoptosisCell culturePyrimidineStereochemistryBiochemistrySignal transductionIn vitroBiologyNursingGeneticsMedicineCell Adhesion Molecules ResearchMelanoma and MAPK PathwaysHER2/EGFR in Cancer Research
Discovery of 7H-pyrrolo[2,3-d]pyridine derivatives as potent FAK inhibitors: Design, synthesis, biological evaluation and molecular docking study | Litcius