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Effects of Chrysin and Its Major Conjugated Metabolites Chrysin-7-Sulfate and Chrysin-7-Glucuronide on Cytochrome P450 Enzymes and on OATP, P-gp, BCRP, and MRP2 Transporters

Violetta Mohos, Eszter Fliszár-Nyúl, Orsolya Ungvári, Éva Bakos, Katalin Kuffa, Tímea Bencsik, Balázs Zoltán Zsidó, Csaba Hetényi, Ágnes Telbisz, Csilla Özvegy‐Laczka, Miklós Poór

2020Drug Metabolism and Disposition49 citationsDOIOpen Access PDF

Topics & Concepts

ChrysinChemistryAbcg2GlucuronideBiochemistryPharmacologyCytochrome P450ATP-binding cassette transporterEnzymeMetaboliteTransporterBiologyFlavonoidAntioxidantGeneDrug Transport and Resistance MechanismsFlavonoids in Medical ResearchNatural product bioactivities and synthesis
Effects of Chrysin and Its Major Conjugated Metabolites Chrysin-7-Sulfate and Chrysin-7-Glucuronide on Cytochrome P450 Enzymes and on OATP, P-gp, BCRP, and MRP2 Transporters | Litcius