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Structure based pharmacophore modelling approach for the design of azaindole derivatives as DprE1 inhibitors for tuberculosis

Suma Kb, Ankita Kumari, Diya Shetty, Everlyse Fernandes, Chethan DV, Judy Jays, Manikanta Murahari

2020Journal of Molecular Graphics and Modelling34 citationsDOI

Topics & Concepts

PharmacophoreADMEChemistryDocking (animal)Mycobacterium tuberculosisComputational biologyStereochemistryCombinatorial chemistryBiochemistryBiologyTuberculosisIn vitroMedicinePathologyNursingTuberculosis Research and EpidemiologyBiochemical and Molecular ResearchCancer therapeutics and mechanisms
Structure based pharmacophore modelling approach for the design of azaindole derivatives as DprE1 inhibitors for tuberculosis | Litcius