Discovery of substituted benzyloxy-benzylamine inhibitors of acetyltransferase Eis and their anti-mycobacterial activity
Allan H. Pang, Keith Green, Nishad Thamban Chandrika, Atefeh Garzan, Ankita Punetha, Selina Y. L. Holbrook, Melisa J. Willby, James E. Posey, Oleg V. Tsodikov, Sylvie Garneau‐Tsodikova
Topics & Concepts
ChemistryMycobacterium tuberculosisAcetyltransferaseBenzylamineAminoglycosideMechanism of actionNon-competitive inhibitionBiochemistryEnzymePharmacologyAcetylationTuberculosisAntibioticsIn vitroBiologyGenePathologyMedicineMedicinal chemistryTuberculosis Research and EpidemiologyMycobacterium research and diagnosisCancer therapeutics and mechanisms