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PDE5 and PDE10 inhibition activates cGMP/PKG signaling to block Wnt/β-catenin transcription, cancer cell growth, and tumor immunity

Gary A. Piazza, Antonio Ward, Xi Chen, Yulia Maxuitenko, Alexander B. Coley, Nada S. Aboelella, Donald J. Buchsbaum, Michael R. Boyd, Adam B. Keeton, Gang Zhou

2020Drug Discovery Today64 citationsDOIOpen Access PDF

Topics & Concepts

SulindacWnt signaling pathwayPhosphodiesterasePharmacologyCell growthCancer cellColorectal cancerCancerCancer researchMedicineSignal transductionChemistryBiologyCell biologyInternal medicineEnzymeBiochemistryNonsteroidalPhosphodiesterase function and regulationInflammatory mediators and NSAID effectsMast cells and histamine
PDE5 and PDE10 inhibition activates cGMP/PKG signaling to block Wnt/β-catenin transcription, cancer cell growth, and tumor immunity | Litcius