Pyrimido[1,2-b]indazole derivatives: Selective inhibitors of human monoamine oxidase B with neuroprotective activity
Badr Jismy, Abdelkarim El Qami, Anja Pišlar, Rok Frlan, Janko Kos, Stanislav Gobec, Damijan Knez, Mohamed Abarbri
Topics & Concepts
ChemistryIndazoleMonoamine oxidaseMonoamine oxidase BMonoamine oxidase ANeuroprotectionStereochemistryCombinatorial chemistryDocking (animal)EnzymeBiochemistryPharmacologyNursingMedicineSynthesis and Biological EvaluationQuinazolinone synthesis and applicationsAdenosine and Purinergic Signaling