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Sultam based Carbonic Anhydrase VII inhibitors for the management of neuropathic pain

Özlem Akgül, Elena Lucarini, Lorenzo Di Cesare Mannelli, Carla Ghelardini, Katia D’Ambrosio, Martina Buonanno, Simona Maria Monti, Giuseppina De Simone, Andrea Angeli, Claudiu T. Supuran, Fabrizio Carta

2021European Journal of Medicinal Chemistry22 citationsDOIOpen Access PDF

Topics & Concepts

ChemistryMoietyNeuropathic painCarbonic anhydraseActive siteGene isoformIn vivoStereochemistrySelectivityPharmacologyEnzymeBiochemistryCatalysisMedicineGeneBiotechnologyBiologyEnzyme function and inhibitionSynthesis and Catalytic ReactionsCholinesterase and Neurodegenerative Diseases
Sultam based Carbonic Anhydrase VII inhibitors for the management of neuropathic pain | Litcius