Synthesis of heterocyclic ring-fused analogs of HMG499 as novel degraders of HMG-CoA reductase that lower cholesterol
Xing-Zi Li, Shi‐You Jiang, Guoqiang Li, Qian-Ru Jiang, Juewan Li, Chenchen Li, Yu-Qin Han, Bao‐Liang Song, Xinran Ma, Wei Qi, Wen‐Wei Qiu
Topics & Concepts
ChemistryReductaseHMG-CoA reductaseCholesterolStatinUbiquitinBiochemistryBiosynthesisEnzymePitavastatinGeneDrug Transport and Resistance MechanismsCancer, Lipids, and MetabolismLipoproteins and Cardiovascular Health