Discovery of a SUCNR1 antagonist for potential treatment of diabetic nephropathy: In silico and in vitro studies
Xuting Zhang, Dongxin Lyu, Shanshan Li, Haiming Xiao, Yufan Qiu, Kangwei Xu, Nianhang Chen, Li Deng, Heqing Huang, Ruibo Wu
Topics & Concepts
In silicoDiabetic nephropathyPharmacophoreIn vitroDrug discoveryVirtual screeningChemistryPharmacologyReceptorComputational biologyBiochemistryCell biologyBiologyDiabetes mellitusEndocrinologyGeneReceptor Mechanisms and SignalingPharmacogenetics and Drug MetabolismComputational Drug Discovery Methods