Discovery of novel USP8 inhibitors via Ubiquitin-Rho-110 fluorometric assay based high throughput screening
Jie Han, Yucheng Tian, Liang Yu, Qilin Zhang, Xi Xu, Yichao Zhang, Jubo Wang, Zengyi Ma, Jinlei Bian, Cheng Luo, Hualiang Jiang, Kaixian Chen, Yao Zhao, Zhiyu Li, Hong Ding
Topics & Concepts
Deubiquitinating enzymeUbiquitinChemistryIC50High-throughput screeningDrug discoverySignal transductionBiochemistryCell biologyIn vitroGeneBiologyUbiquitin and proteasome pathwaysCancer-related Molecular PathwaysHistone Deacetylase Inhibitors Research