Discovery of a covalent inhibitor of heat shock protein 90 with antitumor activity that blocks the co-chaperone binding via C-terminal modification
Li Li, Nannan Chen, Dandan Xia, Shicheng Xu, Wei Dai, Yuanyuan Tong, Lei Wang, Zhengyu Jiang, Qidong You, Xiaoli Xu
Topics & Concepts
Hsp90Chaperone (clinical)Covalent bondCDC37Heat shock proteinBiochemistryCell biologyChemistryBiologyOrganic chemistryMedicinePathologyGeneHeat shock proteins researchComputational Drug Discovery Methods