Design, synthesis and biological activity of N-(amino)piperazine-containing benzothiazinones against Mycobacterium tuberculosis
Apeng Wang, Shijie Xu, Yun Chai, Guimin Xia, Bin Wang, Kai Lv, Chao Ma, Dan Wang, Aoyu Wang, Xiaoyu Qin, Mingliang Liu, Yu Lu
Topics & Concepts
PiperazinehERGChemistryMoietyMycobacterium tuberculosisIn vitroToxicityStereochemistryDrugLead compoundEffluxPharmacologyCombinatorial chemistryTuberculosisBiochemistryOrganic chemistryBiologyMedicinePotassium channelPathologyBiophysicsTuberculosis Research and EpidemiologyCancer therapeutics and mechanismsPhenothiazines and Benzothiazines Synthesis and Activities