Identification of Vitamin K3 and its analogues as covalent inhibitors of SARS-CoV-2 3CLpro
Ruyu Wang, Qing Hu, Haonan Wang, Guanghao Zhu, Mengge Wang, Qian Zhang, Yi‐Shu Zhao, Chunyu Li, Yani Zhang, Guang‐Bo Ge, Hongzhuan Chen, Lili Chen
Topics & Concepts
ChemistryIC50Covalent bondBiochemistrySevere acute respiratory syndrome coronavirus 2 (SARS-CoV-2)VitaminPharmacologyStereochemistryDocking (animal)Coronavirus disease 2019 (COVID-19)In vitroBiologyMedicineInfectious disease (medical specialty)Organic chemistryDiseaseNursingPathologyVitamin C and Antioxidants ResearchComputational Drug Discovery MethodsVitamin K Research Studies