Inhibition of a tonic inhibitory conductance in mouse hippocampal neurones by negative allosteric modulators of α5 subunit-containing γ-aminobutyric acid type A receptors: implications for treating cognitive deficits
Marc A. Manzo, Dian-Shi Wang, Winston W. Li, Arsène Pinguelo, M. Oana Popa, Shahin Khodaei, John Atack, Ruth A. Ross, Beverley A. Orser
Topics & Concepts
GABAA receptorInhibitory postsynaptic potentialTonic (physiology)Allosteric regulationGABAA-rho receptorHippocampal formationChemistryPharmacologyReceptorAllosteric modulatorNeurosciencegamma-Aminobutyric acidPostsynaptic CurrentPatch clampBiophysicsBiologyBiochemistryNeuroscience and Neuropharmacology ResearchNicotinic Acetylcholine Receptors StudyNeurotransmitter Receptor Influence on Behavior