Rhodium(<scp>iii</scp>)-catalyzed C–H activation/annulation of <i>N</i>-iminopyridinium ylides with alkynes and diazo compounds
Xiang Li, Ruihong Zhang, Yaoting Qi, Qing Zhao, Tuanli Yao
Abstract
Rh(<sc>iii</sc>)-Catalyzed C–H activation/annulation of <italic>N</italic>-iminopyridinium ylides with alkynes and diazo compounds has been realized for the synthesis of isoquinolones and isocoumarins.
Topics & Concepts
AnnulationChemistryDiazoRhodiumCatalysisIsocoumarinsMedicinal chemistryStereochemistryOrganic chemistryCatalytic C–H Functionalization MethodsSynthesis and Catalytic ReactionsCyclopropane Reaction Mechanisms