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Characterization of unique functionalities in c-Src domains required for osteoclast podosome belt formation

Takuma Matsubara, William N. Addison, Shoichiro Kokabu, Lynn Neff, William C. Horne, Francesca Gori, Roland Baron

2021Journal of Biological Chemistry21 citationsDOIOpen Access PDF

Abstract

osteoclasts; introduction of constitutively activated SFKs revealed that only c-Src and Fyn could restore this process. To identify the key structural domains responsible, we constructed chimeric Src-Hck and Src-Lyn constructs in which the unique, SH3, SH2, or catalytic domains had been swapped. We found that the Src unique, SH3, and kinase domains were each crucial to establish Src functionality. The SH2 domain could however be substituted with Lyn or Hck SH2 domains. Furthermore, we demonstrate that c-Src's functionality is, in part, derived from an SH3-proximal proline-rich domain interaction with c-Cbl, leading to phosphorylation of c-Cbl Tyr700. These data help clarify Src's unique functionality in the organization of the cytoskeleton in osteoclasts, required for efficient bone resorption and explain why c-Src cannot be replaced, in osteoclasts, by other SFKs.

Topics & Concepts

Proto-oncogene tyrosine-protein kinase SrcLYNPodosomeTyrosine-protein kinase CSKSH3 domainFYNOsteoclastBone resorptionCell biologyOsteopetrosisSH2 domainChemistryInvadopodiaSrc family kinasePhosphorylationTyrosine kinaseBiologySignal transductionBiochemistryReceptorCytoskeletonGeneticsImmunologyCellCancer cellCancerBone Metabolism and DiseasesBone health and treatmentsDermatological and Skeletal Disorders