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Optimization of NAMPT activators to achieve in vivo neuroprotective efficacy

Leibo Wang, Minghui Liu, Yumeng Zu, Yao Hong, Chou Wu, Ruoxi Zhang, Weinan Ma, Haigen Lu, Shuang Xi, Yang Liu, Lan Hua, Gelin Wang, Yefeng Tang

2022European Journal of Medicinal Chemistry22 citationsDOIOpen Access PDF

Topics & Concepts

NeuroprotectionNAD+ kinaseActivator (genetics)ChemistryPharmacologyNicotinamide phosphoribosyltransferaseIn vivoToxicityEx vivoEnzymeIn vitroBiochemistryMedicineBiologyReceptorBiotechnologyOrganic chemistrySirtuins and Resveratrol in MedicineAutophagy in Disease and TherapyCalcium signaling and nucleotide metabolism