Discovery of the SMYD3 Inhibitor BAY-6035 Using Thermal Shift Assay (TSA)-Based High-Throughput Screening

Stefan Gradl, H. Steuber, Joerg Weiske, Magda Szewczyk, Norbert Schmees, Stephan Siegel, Detlef Stoeckigt, Clara D. Christ, Fengling Li, Shawna Organ, Megha Abbey, Steven Kennedy, Irene Chau, Viacheslav V. Trush, Dalia Baršytė-Lovejoy, Peter J. Brown, Masoud Vedadi, C.H. Arrowsmith, Manfred Husemann, Volker Badock, Marcus Bauser, Andrea Haegebarth, Ingo V. Hartung, Carlo Stresemann