Enantiopure substituted pyridines as promising antimalarial drug candidates
Guillaume Bentzinger, Etienne Pair, Jean Guillon, Mathieu Marchivie, Catherine Mullié, Patrice Agnamey, Alexandra Dassonville‐Klimpt, Pascal Sonnet
Topics & Concepts
Enantiopure drugChemistrySN2 reactionCombinatorial chemistryEnantioselective synthesisPyridineMefloquineRegioselectivityRacemizationDihydroartemisininAntimalarial AgentStereochemistryPlasmodium falciparumCatalysisArtemisininOrganic chemistryMalariaImmunologyBiologySynthesis and Catalytic ReactionsMalaria Research and ControlHIV/AIDS drug development and treatment