In vitro identification of imidazo[1,2-a]pyrazine-based antileishmanial agents and evaluation of L. major casein kinase 1 inhibition
Marc‐Antoine Bazin, Sandrine Cojean, Fabrice Pagniez, Guillaume Bernadat, Christian Cavé, Isabelle Ourliac‐Garnier, Marie‐Renée Nourrisson, Cathy Morgado, Carine Picot, L Olivier, Blandine Baratte, Thomas Robert, Gérald F. Späth, Najma Rachidi, Stéphane Bach, Philippe M. Loiseau, Patrice Le Pape, Pascal Marchand
Topics & Concepts
ChemistryMiltefosineCasein kinase 1PharmacologyLeishmaniasisAntiparasiticIn vitroPyrazineMechanism of actionKinaseStereochemistryBiochemistryVisceral leishmaniasisImmunologyMedicineProtein kinase APathologyResearch on Leishmaniasis StudiesTrypanosoma species research and implicationsQuinazolinone synthesis and applications