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Small-molecule inhibition of METTL3 as a strategy against myeloid leukaemia

Eliza Yankova, Wesley Blackaby, Mark R. Albertella, Justyna Rak, Étienne De Braekeleer, Georgia Tsagkogeorga, Ewa S. Pilka, Demetrios Aspris, Dan Leggate, Alan G. Hendrick, Natalie Webster, Byron Andrews, Richard Fosbeary, Patrick Guest, Nerea Irigoyen, Maria Eleftheriou, Malgorzata Gozdecka, João M.L. Dias, Andrew J. Bannister, Binje Vick, Irmela Jeremias, George S. Vassiliou, Oliver Rausch, Konstantinos Tzelepis, Tony Kouzarides

2021Nature1,339 citationsDOIOpen Access PDF

Topics & Concepts

Cancer researchMethyltransferaseIn vivoRNAMyeloid leukemiaBiologyChemistryCell biologyBiochemistryGeneGeneticsMethylationRNA modifications and cancerCancer-related gene regulationRNA Research and Splicing
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