Small-molecule inhibition of METTL3 as a strategy against myeloid leukaemia
Eliza Yankova, Wesley Blackaby, Mark R. Albertella, Justyna Rak, Étienne De Braekeleer, Georgia Tsagkogeorga, Ewa S. Pilka, Demetrios Aspris, Dan Leggate, Alan G. Hendrick, Natalie Webster, Byron Andrews, Richard Fosbeary, Patrick Guest, Nerea Irigoyen, Maria Eleftheriou, Malgorzata Gozdecka, João M.L. Dias, Andrew J. Bannister, Binje Vick, Irmela Jeremias, George S. Vassiliou, Oliver Rausch, Konstantinos Tzelepis, Tony Kouzarides
Topics & Concepts
Cancer researchMethyltransferaseIn vivoRNAMyeloid leukemiaBiologyChemistryCell biologyBiochemistryGeneGeneticsMethylationRNA modifications and cancerCancer-related gene regulationRNA Research and Splicing