Design, synthesis, and mechanism study of dimerized phenylalanine derivatives as novel HIV-1 capsid inhibitors
Xujie Zhang, Lin Sun, Megan E. Meuser, Waleed A. Zalloum, Shujing Xu, Tianguang Huang, Srinivasulu Cherukupalli, Xiangyi Jiang, Xiao Ding, Yucen Tao, Dongwei Kang, Erik De Clercq, Christophe Pannecouque, Alexej Dick, Simon Cocklin, Xinyong Liu, Peng Zhan
Topics & Concepts
ChemistryCapsidStereochemistryPhenylalanineLinkerViral life cycleCombinatorial chemistryBiochemistryAmino acidRNAComputer scienceGeneOperating systemHIV Research and TreatmentHIV/AIDS drug development and treatmentRNA and protein synthesis mechanisms