A potent GPX4 degrader to induce ferroptosis in HT1080 cells
Haoze Song, Jing Liang, Yuanyuan Guo, Yang Liu, Kuiru Sa, Guohong Yan, Wenyan Xu, Wei Xu, Lixia Chen, Hua Li
Topics & Concepts
ChemistryGPX4ProteasomeBiochemistryUbiquitinHT1080Ubiquitin ligaseTernary complexCell biologyGlutathioneGlutathione peroxidaseEnzymeIn vitroBiologyGenePeptidase Inhibition and AnalysisProtein Degradation and InhibitorsHistone Deacetylase Inhibitors Research