Exploring the 1,3-benzoxazine chemotype for cannabinoid receptor 2 as a promising anti-cancer therapeutic
Nicola Gambacorta, Valeria Gasperi, Tatiana Guzzo, Francesco Saverio Di Leva, Fulvio Ciriaco, Cristina Sánchez, Valentina Tullio, Diego Rozzi, Luciana Marinelli, Alessandra Topai, Orazio Nicolotti, Mauro Maccarrone
Topics & Concepts
Cannabinoid receptorChemistryCannabinoid receptor type 2AgonistCannabinoidEndocannabinoid systemMAPK/ERK pathwayPharmacologyAM251ReceptorKinaseSignal transductionCannabinoid Receptor AgonistsBiochemistryBiologyCannabis and Cannabinoid ResearchPhenothiazines and Benzothiazines Synthesis and ActivitiesNeuroscience and Neuropharmacology Research