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Discovery and characterization of novel potent BCR-ABL degraders by conjugating allosteric inhibitor

Haixia Liu, Qianglong Mi, Xinyu Ding, Chencen Lin, Linyi Liu, Chaowei Ren, ShuTing Shen, Yubao Shao, Jinju Chen, Yongqi Zhou, Liting Ji, Heqiao Zhang, Fang Bai, Xiaobao Yang, Qianqian Yin, Biao Jiang

2022European Journal of Medicinal Chemistry29 citationsDOIOpen Access PDF

Topics & Concepts

Chemistrybreakpoint cluster regionPonatinibK562 cellsAllosteric regulationCancer researchABLFusion proteinIbrutinibMutantTyrosine kinaseMutationLeukemiaBiologyGeneticsBiochemistryDasatinibSignal transductionReceptorCellChronic lymphocytic leukemiaGeneRecombinant DNAProtein Degradation and InhibitorsMultiple Myeloma Research and TreatmentsPeptidase Inhibition and Analysis
Discovery and characterization of novel potent BCR-ABL degraders by conjugating allosteric inhibitor | Litcius