Discovery of GPX4 inhibitors through FP-based high-throughput screening
Yu Cao, Bin Wu, Ying Xu, Mingchen Wang, Xinyu Wu, Xiaochen Liang, Jin Lin, Zhihai Li, Hua Lin, Cheng Luo, Shijie Chen, Shijie Chen
Topics & Concepts
ChemistryGPX4SelenocysteinePhospholipid-hydroperoxide glutathione peroxidaseBiochemistrySelenoproteinGlutathione peroxidaseGlutathioneEnzymeCysteineFerroptosis and cancer prognosisCancer, Lipids, and MetabolismInflammatory mediators and NSAID effects