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CuF<sub>2</sub>/DMAP-Catalyzed N-Vinylation: Scope and Mechanistic Study

Krishanu Mondal, Susanta Patra, Pallabi Halder, Narottam Mukhopadhyay, Parthasarathi Das

2022Organic Letters27 citationsDOI

Abstract

CuF2/DMAP has been established as an excellent catalytic system for vinylsilane-promoted N-vinylation of amides and azoles at room temperature without an external fluoride source. A mechanism has been proposed on the basis of the isolation of reactive intermediate [Cu(DMAP)4Cl2], fluoride ion-assisted transmetalation, and ultraviolet–visible spectroscopic studies. The catalytic efficiency of the synthesized and structurally characterized [Cu(DMAP)4Cl2] complex has been demonstrated. The valuable monomers for water-soluble polymers, viz., NVP, NVC, and NVIBA, were synthesized on a gram scale.

Topics & Concepts

ChemistryCatalysisTransmetalationFluorideMonomerCombinatorial chemistryPolymer chemistryPolymerPhotochemistryOrganic chemistryInorganic chemistryChemical Synthesis and AnalysisFluorine in Organic ChemistryAsymmetric Hydrogenation and Catalysis