Targeting focal adhesion kinase (FAK) for cancer therapy: FAK inhibitors, FAK-based dual-target inhibitors and PROTAC degraders
Ming Yang, Hua Xiang, Guoshun Luo
Topics & Concepts
Focal adhesionCancer researchProtein kinase domainDrug discoveryTyrosine kinaseSignal transductionPTK2KinaseTargeted therapyCell biologyBiologyCancerMedicineBioinformaticsProtein kinase ABiochemistryInternal medicineMutantGeneMitogen-activated protein kinase kinaseProtein Degradation and InhibitorsUbiquitin and proteasome pathwaysPeptidase Inhibition and Analysis