LB0005 ORELABRUTINIB, AN IRREVERSIBLE INHIBITOR OF BRUTON'S TYROSINE KINASE (BTK), FOR THE TREATMENT OF SYSTEMIC LUPUS ERYTHEMATOSUS (SLE): RESULTS OF A RANDOMIZED, DOUBLE-BLIND, PLACEBO-CONTROLLED, PHASE IB/IIA DOSE-FINDING STUDY
R. Li, X. Zhu, S. Liu, X. Zhang, C. Xie, Z. Fu, Anaoxue Huang, L. Sun, D. Liu, Jingrun Zhao, Laifeng Wu, Z. Qin, S. Li, Y. Liu, Z. Li
Topics & Concepts
MedicinePlaceboTolerabilityInternal medicineAdverse effectGastroenterologyBruton's tyrosine kinaseNeutropeniaSystemic lupus erythematosusCmaxRandomized controlled trialLupus nephritisPharmacodynamicsPharmacokineticsChemotherapyTyrosine kinaseDiseasePathologyAlternative medicineReceptorChronic Lymphocytic Leukemia ResearchPI3K/AKT/mTOR signaling in cancerRenal Diseases and Glomerulopathies