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Tumor-targeted PROTAC prodrug nanoplatform enables precise protein degradation and combination cancer therapy

Zhifeng Zou, Lei Yang, Hui‐Jun Nie, Jing Gao, Shumin Lei, Yi Lai, Fan Zhang, Ernst Wagner, Haijun Yu, Xiaohua Chen, Zhiai Xu

2024Acta Pharmacologica Sinica48 citationsDOIOpen Access PDF

Topics & Concepts

ProdrugProtein degradationCereblonCancer researchPharmacologyTargeted therapyCancerMedicineChemistryUbiquitinUbiquitin ligaseBiochemistryInternal medicineGeneProtein Degradation and InhibitorsUbiquitin and proteasome pathwaysMultiple Myeloma Research and Treatments
Tumor-targeted PROTAC prodrug nanoplatform enables precise protein degradation and combination cancer therapy | Litcius